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1. Newly Approved Drug Therapies (877) Lunesta (eszopiclone), Sepracor, ...cyclopyrrolone class. It is the S-isomer of the marketed non-benzodiazepine rapid-acting hypnotic zopiclone. Lunesta raises levels of an amino acid called Gamma-Aminobutyric Acid (GABA). GABA slows down ......sleep. Literature References Drug Enforcement Administration, Department of Justice. Schedules of controlled substances: placement of Zopiclone into schedule IV. Final rule. Fed Regist. 2005 Apr 4;70(63):16935-7. Eszopiclone ...View Page
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